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Bpsbioscience/HSP90α C-Terminal Domain TR-FRET Assay Kit/50289/96 reactions

Description:
ThisassaykitisdesignedtomeasuretheinhibitionoftheHSP90αbindingtoitsproteintargetPPID(alsoknownasCyclophilinD)inahomogeneous,96reactionformat.Thisassayrequiresnotime-consumingwashingsteps,makingitespeciallysuitableforhighthroughputscreeningapplications.Theassayprocedureisstraightforwardandsimple.Asamplecontainingterbium-labeleddonor,dye-labeledacceptor,HSP90α,substrate,andaninhibitorisincubatedfor2hours.Theprotein-proteininteractionisthenassayedbymeasuringtheTR-FRETbetweenthePPIDandHSP90αusingafluorescencereader.
Synonym(s):
HSP90,Assaykit,HSP90a,HSP90α,Fretassaykit
Format:

COMPONENTS:

Instructionsforuse:
Seeassaykitdatasheetfordetailedprotocol
Storage/StABIlity:
Atleast6monthsfromdateofreceiptwhenstoredasdirected.
Application(s):
GreatforscreeningsmallmolecularinhibitorsfordrugdiscoveryandHTSapplications.
Reference(s):
Allan,R.K.etal.J.Biol.Chem2006281(11):7161-71
Warning(s):
Avoidfreeze/thawcycles.
ScientificCategory:
HeatShockProteins
ProductType:
AssayKit
Datashownislot-specific.Contactusforspecificinformationonotherlots.
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