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Anatrace//MCSG1/MCSG1-2 100 ML

Selective inhibitor of Usp14 (IC50<4 µM). Enhances proteasome activity and substrate proteolysis1,2. Inhibits Dengue virus replication3. In prion-infected CAD5 cells activation of the ubiquitin proteasome system by IU1 is sufficient to induce clearance of polyubiquitinated substrates and reduce misfolded prion protein load4. Attenuates ischemia/reperfusion-induced neuronal injury in a mouse model5. Cell permeable.
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