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ArelativelypotentMT2melatoninreceptorantagonist(pKivalue=8.03),displaying89-and229-foldselectivityoverMT1andGPR50(melatonin-relatedorphanreceptor)respectively.
DH97isalsoofferedaspartoftheTocriscreenPlus.FindoutmoreaboutcompoundlibrariesavailablefromTocris.
| M.Wt | 334.46 |
| Formula | C22H26N2O |
| Storage | StoreatRT |
| CASNumber | 220339-00-4 |
| PubChemID | 3467177 |
| InChIKey | HDOIPCLEKCEANF-UHFFFAOYSA-N |
| Smiles | CCCCC(=O)NCCC1=C(CC2=CC=CC=C2)NC2=CC=CC=C12 |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
| Solubility | Solubleto100mMinDMSO |
Thefollowingdataisbasedontheproductmolecularweight334.46.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.99mL | 14.95mL | 29.9mL |
| 5mM | 0.6mL | 2.99mL | 5.98mL |
| 10mM | 0.3mL | 1.49mL | 2.99mL |
| 50mM | 0.06mL | 0.3mL | 0.6mL |