Potent,selectiveGABABreceptorantagonist(IC50=85nM).
SoldwiththepermissionofNovartisPharmaAG
| M.Wt | 384.24 |
| Formula | C15H24Cl2NO4P |
| Storage | Desiccateat+4°C |
| Purity | ≥98%(HPLC) |
| CASNumber | 139667-74-6 |
| PubChemID | 132252 |
| InChIKey | GJZVQXWEIYRHBE-UHFFFAOYSA-N |
| Smiles | ClC1=CC=C(CNCCCP(C(OCC)OCC)(O)=O)C=C1Cl |
Thetechnicaldataprovidedaboveisforguidanceonly.ForbatchspecificdatarefertotheCertificateofAnalysis.
AllTocrisproductsareintendedforlaboratoryresearchuseonly.
| Solvent | MaxConc.mg/mL | MaxConc.mM | |
|---|---|---|---|
| Solubility | |||
| water | 3.84 | 10mMwithsonication |
Thefollowingdataisbasedontheproductmolecularweight384.24.Batchspecificmolecularweightsmayvaryfrombatchtobatchduetosolventofhydration,whichwillaffectthesolventvolumesrequiredtopreparestocksolutions.
| Concentration/SolventVolume/Mass | 1mg | 5mg | 10mg |
|---|---|---|---|
| 1mM | 2.6mL | 13.01mL | 26.03mL |
| 5mM | 0.52mL | 2.6mL | 5.21mL |
| 10mM | 0.26mL | 1.3mL | 2.6mL |
| 50mM | 0.05mL | 0.26mL | 0.52mL |