Functionalizedvon-Hippel-Lindauproteinligand(VHL)forPROTACresearchanddevelopment;incorporatesanE3ligaseligandplusashortalkyllinkerreadyforconjugationtoatargetproteinligand.PartofarangeoffunctionalizedtoolmoleculesforPROTACR&D.
Application
FunctionalizedVHLligandforPROTACs;incorporatesanE3ligaseligandplusashortalkyllinker.
ProductInformation
Purity: >95%
MW: 566.16
Formula: C27H39N5O4S.HCl
PhysicalState: Lyophilizedwhitesolid
Quantity: 5mg;10mg;25mg
Solubility: 50mg/mLinDMSO;50mg/mLinwater
Storage: Storeat-20C.
Documents
References
1. Salami etal (2017)Wastedisposal-Anattractivestrategyforcancertherapy.Science 355 1163PMID: 28302825
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